Cyclopropanemethanamine → HCID 59568470, compound

Participants

Reaction Steps

As described for example 163c, 3-((3-(5-fluoropyridin-2-yl)-5-methylisoxazol-4-yl)methylamino)-1-methyl-1H-pyrazole-5-carboxylic acid (92 mg, 0.28 mol) was converted, using aminomethylcyclopropane instead of isopropylamine, to the title compound (85 mg, 80%) which was obtained as a white solid. MS: m/e=385.2 [M+H]+.

Provenance & Evidence