Benzyl Alcohol → HCID 178494001, compound

HRID 1704760Notes

Reaction equation

HRID 1704760 reaction equation
[CH3:1][O:2]C1C2C=NC3NN=CC=3C=2N2N=CN=C2N=1.Cl[C:20]1[C:25]2[CH:26]=[N:27][C:28]3[N:32](CC)[N:31]=[CH:30][C:29]=3[C:24]=2[N:23]2[N:35]=[CH:36][N:37]=[C:22]2[N:21]=1.C(O)[C:39]1[CH:44]=[CH:43][CH:42]=[CH:41][CH:40]=1>C(O)C>[C:39]1([C:20]2[C:25]3[CH:26]=[N:27][C:28]4[NH:32][N:31]=[CH:30][C:29]=4[C:24]=3[N:23]3[N:35]=[C:36]([O:2][CH3:1])[N:37]=[C:22]3[N:21]=2)[CH:44]=[CH:43][CH:42]=[CH:41][CH:40]=1

Participants

5

Reactant 3

HCID 244Benzyl AlcoholHCID 227584865-Chloro-8-ethyl-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]-triazolo[1,5-a]pyrimidineHCID 178494003HCID 178494003, compound

Product 1

HCID 178494001HCID 178494001, compound

Reagents, catalysts & solvents 1

HCID 702EthanolSolvent

Procedure

By substituting the 5-chloro-8H-pyrazolo[4',3':5,6]-pyrido[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine of Example 15 for the 5-chloro-8-ethyl-8H-pyrazolo[4',3':5,6]pyrido-[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine and benzyl alcohol for the ethanol in the procedure of Example 4, 5-phenyl-methoxy-8H-pyrazolo[4',3':5,6]pyrido[3,4-e][1,2,4]triazolo[1,5-a]pyrimidine is obtained.

Sources & evidence

ORD record
ord-06845e9e69eb4eb1b0668a890c14e8ae
Source dataset
uspto-grants-1978_11
Patent number
US04127655

Reaction notes

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