4-Bromopyridinium chloride → HCID 4184629, compound
Reaction equation
Cl.Br[C:3]1[CH:8]=[CH:7][N:6]=[CH:5][CH:4]=1.[C:9]([C:11]1[CH:16]=[CH:15][C:14](B(O)O)=[CH:13][CH:12]=1)#[N:10]>>[N:6]1[CH:7]=[CH:8][C:3]([C:14]2[CH:15]=[CH:16][C:11]([C:9]#[N:10])=[CH:12][CH:13]=2)=[CH:4][CH:5]=1Participants
3
Procedure
The title compound was prepared in a similar manner to that described in Reference Example 11 using 4-bromopyridine hydrochloride instead of 1-bromo-3-pentyloxybenzene and 4-cyanophenylboronic acid instead of tert-butyl N-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolane-2-yl)-benzyl]carbamate.
Sources & evidence
- ORD record
- ord-288140bf12de404baaa107315358407d
- Source dataset
- uspto-grants-2010_09
- Patent number
- US07795236B2
Reaction notes
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