(3-hydroxyphenyl)boronic Acid → HCID 58911434, compound

HRID 1713310Notes

Reaction equation

HRID 1713310 reaction equation
Br[C:2]1[CH:3]=[C:4]([CH:14]=[CH:15][CH:16]=1)[CH2:5][NH:6][C:7](=[O:13])[O:8][C:9]([CH3:12])([CH3:11])[CH3:10].[OH:17][C:18]1[CH:19]=[C:20](B(O)O)[CH:21]=[CH:22][CH:23]=1>>[OH:17][C:18]1[CH:23]=[C:22]([C:2]2[CH:16]=[CH:15][CH:14]=[C:4]([CH2:5][NH:6][C:7](=[O:13])[O:8][C:9]([CH3:12])([CH3:11])[CH3:10])[CH:3]=2)[CH:21]=[CH:20][CH:19]=1

Participants

3

Reactant 2

HCID 2734359(3-hydroxyphenyl)boronic AcidHCID 11033439tert-Butyl 3-bromobenzylcarbamate

Product 1

HCID 58911434HCID 58911434, compound

Procedure

The title compound was prepared in a similar manner to that described in Reference Example 2 using tert-butyl N-(3-bromobenzyl)carbamate instead of tert-butyl N-(4-bromobenzyl)carbamate and 3-hydroxyphenylboronic acid instead of 3-benzyloxyphenylboronic acid.

Sources & evidence

ORD record
ord-a2b70ad3352a496faa70ba3f6d54d0a5
Source dataset
uspto-grants-2010_09
Patent number
US07795236B2

Reaction notes

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