5-Bromo-2-methyl-4-(4-nitrophenyl)-1,3-oxazole → 4-[2-methyl-4-(4-nitrophenyl)-1,3-oxazol-5-yl]-1-[(4-methylphenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridine

Participants

Role	Name	HCID	Charge
Reactant	5-Bromo-2-methyl-4-(4-nitrophenyl)-1,3-oxazole	HCID 21787037	—
Reactant	1-Tosyl-1H-pyrrolo(2,3-B)pyridine-4-boronic acid pinacol ester	HCID 49758926	—
Product	4-[2-methyl-4-(4-nitrophenyl)-1,3-oxazol-5-yl]-1-[(4-methylphenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridine	HCID 69000494	—

Reaction Steps

Following the procedure described for Intermediate 6 with 5-bromo-2-methyl-4-(4-nitrophenyl)-1,3-oxazole and [(4-methylphenyl)sulfonyl]-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrrolo[2,3-b]pyridine provided the title compound. ESMS [M+H]+: 476.2

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US07495102B2
Source dataset	uspto-grants-2009_02
ORD ID	ord-d0107e43fd234e9ca2ecbd02a172db37
Source note	uspto-grants-2009_02