2-Amino-3-benzyloxypyridine → HCID 19016496, compound

HRID 1728597Notes

Reaction equation

HRID 1728597 reaction equation
[NH2:1][C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[N:7]([CH3:11])[CH:6]=[CH:5]2.[C:12](C1NC=CN=1)(C1NC=CN=1)=[O:13].[NH2:24][C:25]1[C:30]([O:31][CH2:32][C:33]2[CH:38]=[CH:37][CH:36]=[CH:35][CH:34]=2)=[CH:29][CH:28]=[CH:27][N:26]=1>>[CH3:11][N:7]1[C:8]2[C:4](=[CH:3][C:2]([NH:1][C:12]([NH:24][C:25]3[C:30]([O:31][CH2:32][C:33]4[CH:34]=[CH:35][CH:36]=[CH:37][CH:38]=4)=[CH:29][CH:28]=[CH:27][N:26]=3)=[O:13])=[CH:10][CH:9]=2)[CH:5]=[CH:6]1

Participants

4

Reactant 3

HCID 903342-Amino-3-benzyloxypyridineHCID 27695641-methyl-1H-indol-5-amineHCID 5250894Bis-(1H-imidazol-2-YL)-methanone

Product 1

HCID 19016496HCID 19016496, compound

Procedure

The title compound was prepared from 5-amino-1-methyl-1H-indole (D3), carbonyl diimidazole and 2-amino-3-benzyloxypyridine using a procedure similar to that described in Example 1.

Sources & evidence

ORD record
ord-25ddb1b0ffe74b5bb6053b132e9279e8
Source dataset
uspto-grants-1994_07
Patent number
US05328922

Reaction notes

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