HCID 495677, compound → HCID 19011701, compound

HRID 1729215Notes

Reaction equation

HRID 1729215 reaction equation
O[CH:2]1CN(C(=O)C2C=CC3OCOC=3C=2)C(C(O)=O)C1.[OH:21][CH:22]1[CH2:26][N:25]([C:27](=[O:40])[C:28]2[CH:33]=[C:32]([O:34][CH3:35])[C:31]([O:36][CH3:37])=[C:30]([O:38][CH3:39])[CH:29]=2)[CH:24]([C:41]([OH:43])=[O:42])[CH2:23]1>>[CH3:2][O:42][C:41]([CH:24]1[CH2:23][CH:22]([OH:21])[CH2:26][N:25]1[C:27](=[O:40])[C:28]1[CH:29]=[C:30]([O:38][CH3:39])[C:31]([O:36][CH3:37])=[C:32]([O:34][CH3:35])[CH:33]=1)=[O:43]

Participants

3

Reactant 2

HCID 495677HCID 495677, compoundHCID 16771157HCID 16771157, compound

Product 1

HCID 19011701HCID 19011701, compoundYield 40%

Procedure

By carrying out the procedure as in Example 11, but replacing 4-hydroxy-1-(3,4-methylenedioxybenzoyl)pyrrolidine-2-carboxylic acid by the 4-hydroxy-1-(3,4,5-trimethoxybenzoyl)pyrrolidine-2-carboxylic acid obtained in Example 8, the title product is obtained.

Sources & evidence

ORD record
ord-ba0f809be763405995a5c76979bccc8f
Source dataset
uspto-grants-1994_07
Patent number
US05332735

Reaction notes

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