HCID 21495095, compound → HCID 21495092, compound

HRID 1731121Notes

Reaction equation

HRID 1731121 reaction equation
N1C2=CN=NC2=[CH:4]N=N1.[C:10]([NH:13][C:14]1[N:19]2[N:20]=[CH:21][C:22]([C:23]3[CH:28]=[CH:27][N:26]=[CH:25]N=3)=[C:18]2[N:17]=[CH:16][N:15]=1)(=[O:12])[CH3:11].C(NC1N2N=CC(C3C=NC=CN=3)=C2N=CN=1)(=O)C>>[C:10]([NH:13][C:14]1[N:19]2[N:20]=[CH:21][C:22]([C:23]3[CH:28]=[CH:27][N:26]=[CH:25][CH:4]=3)=[C:18]2[N:17]=[CH:16][N:15]=1)(=[O:12])[CH3:11]

Participants

4

Reactant 3

HCID 21495095HCID 21495095, compoundHCID 21495102HCID 21495102, compoundHCID 178420931HCID 178420931, compound

Product 1

HCID 21495092HCID 21495092, compound

Procedure

By replacing the pyrazolotriazine employed in Example 4 by an equivalent quantity of the end product of Example 2 or Example 3 there is obtained, respectively, 4-acetamido-8-(4-pyrimidinyl)-pyrazolo-[1,5-a][1,3,5]triazine and 4-acetamido-8-(2-pyrazinyl)-pyrazolo[1,5-a][1,3,5]triazine.

Workup

  1. customExample 3 there is obtained

Sources & evidence

ORD record
ord-61a629a6440d47d39b1c29c494155ea2
Source dataset
uspto-grants-1976_11
Patent number
US03995039

Reaction notes

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