Sodium borohydride → HCID 57195349, compound

Participants

Reaction Steps

235 mg (0.378 mmol) of (2R*,4S*)-2-benzyl-1-(diphenylacetyl)-N-(4-quinolylmethyl)-N-trifluoroacetyl-4-piperidinamine are reacted with 58 mg (1.51 mmol) of sodium borohydride in analogy to Example 2. The title compound ##STR43## is obtained as white foam. TLC: methylene chloride/methanol/conc. ammonia (700:50:1) Rf =0.49, FD-MS: M+ =525.

Provenance & Evidence