HuagongsheHuagongshe Chemistry Print Report · For research reference only
6-benzyloxy-3-amino-1,2,3,4-tetrahydro-9H-carbazole → 6-benzyloxy-3-(2-(1-isopropyl-1H-pyrazol-4-yl)ethyl)amino-1,2,3,4-tetrahydro-9H-carbazole
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 6-benzyloxy-3-amino-1,2,3,4-tetrahydro-9H-carbazole | HCID 22611308 | — |
| Reactant | 2-(1-isopropyl-1H-pyrazol-4-yl)-1-mesyloxyethane | HCID 22611512 | — |
| Product | 6-benzyloxy-3-(2-(1-isopropyl-1H-pyrazol-4-yl)ethyl)amino-1,2,3,4-tetrahydro-9H-carbazole | HCID 22611185 | 63.4% |
Reaction Steps
Beginning with 0.698 gm (2.39 mMol) 6-benzyloxy-3-amino-1,2,3,4-tetrahydro-9H-carbazole and 0.787 gm (3.39 mMol) 2-(1-isopropyl-1H-pyrazol-4-yl)-1-mesyloxyethane, 0.649 gm (63.4%) of the desired compound were prepared by the procedure described in detail in EXAMPLE B-72.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US05962473 |
| Source dataset | uspto-grants-1999_10 |
| ORD ID | ord-5885377232b04635a660f65eb10e6d98 |
| Source note | uspto-grants-1999_10 |