5-Bromoindole → HCID 19390954, compound

HRID 1756652Notes

Reaction equation

HRID 1756652 reaction equation
[NH2:1][C:2]1[N:6]([C:7]2[CH:8]=[C:9](B3OCCCO3)[CH:10]=[CH:11][CH:12]=2)[C:5]2[CH:19]=[CH:20][CH:21]=[CH:22][C:4]=2[N:3]=1.Br[C:24]1[CH:25]=[C:26]2[C:30](=[CH:31][CH:32]=1)[NH:29][CH:28]=[CH:27]2>>[NH2:1][C:2]1[N:6]([C:7]2[CH:12]=[CH:11][CH:10]=[C:9]([C:24]3[CH:25]=[C:26]4[C:30](=[CH:31][CH:32]=3)[NH:29][CH:28]=[CH:27]4)[CH:8]=2)[C:5]2[CH:19]=[CH:20][CH:21]=[CH:22][C:4]=2[N:3]=1

Participants

3

Reactant 2

HCID 249055-BromoindoleHCID 185220553-(2-Amino-1-benzimidazolyl)-phenyl-1,3,2-dioxaborinane

Product 1

HCID 19390954HCID 19390954, compound

Procedure

2-Amino-1-[3-(5-indolyl)phenyl]benzimidazole was prepared from 3-(2-amino-1-benzimidazolyl)-phenyl-1,3,2-dioxaborinane and 5-bromoindole according to method A. mp 120°-123° C.

Sources & evidence

ORD record
ord-0239be96c0d845849ec157a9e3e1d3c8
Source dataset
uspto-grants-1995_08
Patent number
US05441969

Reaction notes

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