4-Carboxyphenylboronic Acid → HCID 67974892, compound

Participants

Reaction Conditions

Reaction Steps

Followed the coupling procedure described for Example 3, starting from 1-chloro-6-methoxynaphthalen-2-yl trifluoromethanesulfonate (Intermediate 4, 1 equiv) and 4-boronobenzoic acid (1.2 equiv), where the mixture was stirred at 80° C. for 2 hours. The crude product was obtained after workup and was taken on without purification.

Provenance & Evidence