(3S)-3-methylmorpholine → HCID 67382589, compound

HRID 1771538Notes

Reaction equation

HRID 1771538 reaction equation
[CH:1]12[O:8][CH:5](CC1)[CH2:4][N:3]([C:9]1[N:14]=[C:13]([C:15]3[CH:21]=[CH:20][C:18]([NH2:19])=[CH:17][CH:16]=3)[CH:12]=[CH:11][N:10]=1)[CH2:2]2.[CH3:22][C@H]1COCCN1>>[CH3:22][C@@H:4]1[N:3]([C:9]2[N:14]=[C:13]([C:15]3[CH:16]=[CH:17][C:18]([NH2:19])=[CH:20][CH:21]=3)[CH:12]=[CH:11][N:10]=2)[CH2:2][CH2:1][O:8][CH2:5]1

Participants

3

Reactant 2

HCID 12012220(3S)-3-methylmorpholineHCID 67382726HCID 67382726, compound

Product 1

HCID 67382589HCID 67382589, compound

Procedure

Method as described for intermediate 26 using (S)-3-methylmorpholine. (699 mg, 95%).

Sources & evidence

ORD record
ord-03daf12455084611bc937cfaa7aa8068
Source dataset
uspto-grants-2016_02
Patent number
US09249129B2

Reaction notes

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