2-Phenylpyridine-3-boronic acid → HCID 86296579, compound

HRID 1773671Notes

Reaction equation

HRID 1773671 reaction equation
[C:1]1([C:7]2[C:12](B(O)O)=[CH:11][CH:10]=[CH:9][N:8]=2)[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1.[CH3:16][C:17]1[C:21]([C:22]2[CH:23]=[C:24](C3C(C)=CC=C4C=3C=CC=N4)[C:25]3[O:29][C:28](=[O:30])[NH:27][C:26]=3[CH:31]=2)=[C:20]([CH3:43])[O:19][N:18]=1>>[CH3:16][C:17]1[C:21]([C:22]2[CH:23]=[C:24]([C:12]3[C:7]([C:1]4[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=4)=[N:8][CH:9]=[CH:10][CH:11]=3)[C:25]3[O:29][C:28](=[O:30])[NH:27][C:26]=3[CH:31]=2)=[C:20]([CH3:43])[O:19][N:18]=1

Participants

3

Reactant 2

HCID 27630852-Phenylpyridine-3-boronic acidHCID 86296578HCID 86296578, compound

Product 1

HCID 86296579HCID 86296579, compound

Procedure

The title compound was synthesized using 2-phenylpyridin-3-ylboronic acid in a similar fashion with 5-(3,5-dimethylisoxazol-4-yl)-7-(6-methylquinolin-5-yl)benzo[d]oxazol-2(3H)-one (Example 11).

Sources & evidence

ORD record
ord-c20edad371de4aeb9cb2dfc16f61b414
Source dataset
uspto-grants-2016_02
Patent number
US09255089B2

Reaction notes

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