(Pyridin-4-yl)boronic acid → HCID 5275995, compound

HRID 1788431Notes

Reaction equation

HRID 1788431 reaction equation
ClC1[CH:41]=[CH:40][C:5]([C:6]2[C:11]([C:12]3[CH:21]=[CH:20][C:19]4[C:14](=[CH:15][CH:16]=[C:17]([C:22]5[N:26]([CH:27]6[CH2:32][CH2:31][CH2:30][CH2:29][CH2:28]6)[C:25]6[CH:33]=[CH:34][C:35]([C:37]([OH:39])=[O:38])=[CH:36][C:24]=6[N:23]=5)[CH:18]=4)[N:13]=3)=[CH:10][CH:9]=[CH:8][CH:7]=2)=[CH:4][CH:3]=1.[N:42]1C=CC(B(O)O)=CC=1>>[CH:27]1([N:26]2[C:25]3[CH:33]=[CH:34][C:35]([C:37]([OH:39])=[O:38])=[CH:36][C:24]=3[N:23]=[C:22]2[C:17]2[CH:16]=[C:15]3[C:14](=[CH:19][CH:18]=2)[N:13]=[C:12]([C:11]2[CH:10]=[CH:9][CH:8]=[CH:7][C:6]=2[C:5]2[CH:4]=[CH:3][N:42]=[CH:41][CH:40]=2)[CH:21]=[CH:20]3)[CH2:28][CH2:29][CH2:30][CH2:31][CH2:32]1

Participants

3

Reactant 2

HCID 2734379(Pyridin-4-yl)boronic acidHCID 5276010HCID 5276010, compound

Product 1

HCID 5275995HCID 5275995, compound

Procedure

The title compound was synthesized as described for Compound 387 except pyridine-4-boronic acid was used instead of 4-chlorophenyl-boronic acid.

Sources & evidence

ORD record
ord-8e17b79c8d794eb18eacc939146659d4
Source dataset
uspto-grants-2009_03
Patent number
US07511145B2

Reaction notes

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