HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-Amino-1-(3-phenyl-1,2,4-oxadiazol-5-yl)-butan-1-ol → (r)-4,4-Dimethyl-2-(2-morpholin-4-yl-2-oxo-ethyl)-5-phenyl-pentanoic acid[1-(3-phenyl-1,2,4-oxadiazole-5-carbonyl)-propyl]-amide
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-Amino-1-(3-phenyl-1,2,4-oxadiazol-5-yl)-butan-1-ol | HCID 21962745 | — |
| Reactant | (R)-4,4-Dimethyl-2-(2-morpholin-4-yl-2-oxo-ethyl)-5-phenyl-pentanoic acid | HCID 58619484 | — |
| Product | (r)-4,4-Dimethyl-2-(2-morpholin-4-yl-2-oxo-ethyl)-5-phenyl-pentanoic acid[1-(3-phenyl-1,2,4-oxadiazole-5-carbonyl)-propyl]-amide | HCID 58619496 | — |
Reaction Steps
It is similarly prepared (as mixture of diastereoisomers) according to general procedure given for example 10 above but using (R)-4,4-Dimethyl-2-(2-morpholin-4-yl-2-oxo-ethyl)-5-phenyl-pentanoic acid and 2-Amino-1-(3-phenyl-1,2,4-oxadiazol-5-yl)-butan-1-ol
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07030116B2 |
| Source dataset | uspto-grants-2006_04 |
| ORD ID | ord-a2b4e0e2865d42efbd5a1cb2b276a200 |
| Source note | uspto-grants-2006_04 |