4-Carboxyphenylboronic Acid → HCID 57475016, compound

HRID 1798440Notes

Reaction equation

HRID 1798440 reaction equation
B([C:4]1[CH:12]=[CH:11][C:7]([C:8]([OH:10])=[O:9])=[CH:6][CH:5]=1)(O)O.Br[C:14]1[CH:15]=[C:16]2[C:21](=[CH:22][CH:23]=1)[O:20][CH:19]=[CH:18][C:17]2=[O:24]>>[O:24]=[C:17]1[C:16]2[C:21](=[CH:22][CH:23]=[C:14]([C:4]3[CH:12]=[CH:11][C:7]([C:8]([OH:10])=[O:9])=[CH:6][CH:5]=3)[CH:15]=2)[O:20][CH:19]=[CH:18]1

Participants

3

Reactant 2

HCID 3121834-Carboxyphenylboronic AcidHCID 5485226-Bromochromone

Product 1

HCID 57475016HCID 57475016, compound

Procedure

The title compound was prepared as described in EXAMPLE 4A using 4-boronobenzoic acid in place of 4-(methoxycarbonyl)phenylboronic acid and 6-bromo-4H-chromen-4-one in place of 1-bromo-3-iodobenzene.

Sources & evidence

ORD record
ord-f56a868e5c4849619d36ecb16827de27
Source dataset
uspto-grants-2013_01
Patent number
US08343967B2

Reaction notes

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