HCID 44135954, compound → HCID 68942993, compound
Reaction equation
CNC1N=C(C2C=CC=CN=2)C=C(C2C=NC=CC=2)C=1[C:21]1[CH:22]=[N:23][N:24]([CH:26]2[CH2:31][CH2:30][NH:29][CH2:28][CH2:27]2)[CH:25]=1.Br[C:33]1[CH:34]=[C:35]([C:39]2[CH:44]=[C:43]([NH:45][CH3:46])[N:42]=[C:41]([C:47]3[CH:52]=[CH:51][CH:50]=[C:49]([CH3:53])[N:48]=3)[CH:40]=2)[CH:36]=[N:37][CH:38]=1>>[CH3:46][NH:45][C:43]1[N:42]=[C:41]([C:47]2[CH:52]=[CH:51][CH:50]=[C:49]([CH3:53])[N:48]=2)[CH:40]=[C:39]([C:35]2[CH:36]=[N:37][CH:38]=[C:33]([C:21]3[CH:22]=[N:23][N:24]([CH:26]4[CH2:31][CH2:30][NH:29][CH2:28][CH2:27]4)[CH:25]=3)[CH:34]=2)[CH:44]=1Participants
3
Procedure
This compound is prepared analogously to Methyl-[5″-(1-piperidin-4-yl-1H-pyrazol-4-yl)-[2,2′;4′,3″]terpyridin-6′-yl]-amine (Example 2.183) by replacing (5″-Bromo-[2,2′;4′,3″]terpyridin-6′-yl)-methyl-amine (Example 2.1, step1) with (5″-Bromo-6-methyl-[2,2′;4′,3″]terpyridin-6′-yl)-methyl-amine (Example 1.27).
Sources & evidence
- ORD record
- ord-c069bbdd98204f028f43b75b8d4c0c47
- Source dataset
- uspto-grants-2013_01
- Patent number
- US08343966B2
Reaction notes
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