Morpholine → HCID 67968025, compound

Participants

Reaction Steps

The product was prepared in the same manner as described in example 4 using 5-(2-(cyclopropyl(methyl)amino)-[1,2,4]triazolo[1,5-a]pyridine-7-ylcarbamoyl)-1-methyl-1H-pyrazole-4-carboxylic acid (70 mg, 197 μmol) and morpholine (68.6 μl, 788 μmol) as starting materials. The reaction affords 2-Methyl-4-(morpholine-4-carbonyl)-2H-pyrazole-3-carboxylic acid [2-(cyclopropyl-methyl-amino)-[1,2,4]triazolo[1,5-a]pyridine-7-yl]-amide (82 mg, 98.1%) as off-white solid. MS: m/z=325.1 (M+H+).

Provenance & Evidence