5-Fluoro-2-methoxyphenylboronic acid → HCID 67238968, compound
Reaction equation
Br[C:2]1[CH:7]=[CH:6][C:5]([S:8]([C:11]2[CH:16]=[CH:15][CH:14]=[C:13]([F:17])[CH:12]=2)(=[O:10])=[O:9])=[C:4]([F:18])[CH:3]=1.[F:19][C:20]1[CH:21]=[CH:22][C:23]([O:29][CH3:30])=[C:24](B(O)O)[CH:25]=1>>[F:17][C:13]1[CH:12]=[C:11]([S:8]([C:5]2[CH:6]=[CH:7][C:2]([C:22]3[CH:21]=[C:20]([F:19])[CH:25]=[CH:24][C:23]=3[O:29][CH3:30])=[CH:3][C:4]=2[F:18])(=[O:10])=[O:9])[CH:16]=[CH:15][CH:14]=1Participants
3
Procedure
The subtitle compound was prepared by the method of example 2 step (ii) using the product of step (ii) and 5-fluoro-2-methoxybenzene boronic acid.
Sources & evidence
- ORD record
- ord-c0f31a801f8144a3ba157e5d2aabbb4f
- Source dataset
- uspto-grants-2013_01
- Patent number
- US08349897B2
Reaction notes
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