HCID 59255049, compound → HCID 59255056, compound

HRID 1809358Notes

Reaction equation

HRID 1809358 reaction equation
[F:1][C:2]1[CH:3]=[C:4]([C:13]([O:15]CC)=[O:14])[C:5](=[O:12])[N:6]([CH:9]([CH3:11])[CH3:10])[C:7]=1[CH3:8].ClC1C=C(C(OCC)=O)C(=O)N(C(C)C)C=1C>>[F:1][C:2]1[CH:3]=[C:4]([C:13]([OH:15])=[O:14])[C:5](=[O:12])[N:6]([CH:9]([CH3:11])[CH3:10])[C:7]=1[CH3:8]

Participants

3

Procedure

The title compound was prepared according to the procedure of Example 1(7), but using ethyl 5-fluoro-1-isopropyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxylate as prepared in 5(1) instead of ethyl 5-chloro-1-isopropyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxylate.

Sources & evidence

ORD record
ord-8275ce9854ff42e4b210620321f6e513
Source dataset
uspto-grants-2013_01
Patent number
US08362038B2

Reaction notes

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