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HRID 1810439作成日：2026年10月25日

3-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-4-bromo-benzoic acid → 2-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-5'-ethoxycarbonylmethyl-2'-methoxy-biphenyl-4-carboxylic acid

https://huagongshe.com/reaction/1810439

反応式

関与物質

役割名称HCID仕込み量
反応物3-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-4-bromo-benzoic acidHCID 57419864—
反応物[4-Methoxy-3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-acetic acid ethyl esterHCID 58120060—
生成物2-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-5'-ethoxycarbonylmethyl-2'-methoxy-biphenyl-4-carboxylic acidHCID 54674329—

反応手順

Prepared according to the procedure described in Example 1, Step 4, using the following starting materials: 3-[(benzyloxycarbonyl-ethyl-amino)-methyl]-4-bromo-benzoic acid and [4-methoxy-3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-acetic acid ethyl ester. M+H is 506.

情報源と証拠

DOI10.6084/m9.figshare.5104873.v1
特許番号US08362044B2
出典データセットuspto-grants-2013_01
ORD IDord-abf51bf68cbe489bad419ffaa20369c6
出典メモuspto-grants-2013_01