Pivaloyl chloride → HCID 57884003, compound

HRID 1817883Notes

Reaction equation

[NH2:1][C:2]1[CH:7]=[C:6]([S:8]([CH:11]([CH3:13])[CH3:12])(=[O:10])=[O:9])[CH:5]=[CH:4][C:3]=1[NH:14][CH2:15][C:16]1([OH:21])[CH2:20][CH2:19][CH2:18][CH2:17]1.[C:22](Cl)(=O)[C:23]([CH3:26])([CH3:25])[CH3:24]>>[C:23]([C:26]1[N:14]([CH2:15][C:16]2([OH:21])[CH2:20][CH2:19][CH2:18][CH2:17]2)[C:3]2[CH:4]=[CH:5][C:6]([S:8]([CH:11]([CH3:12])[CH3:13])(=[O:9])=[O:10])=[CH:7][C:2]=2[N:1]=1)([CH3:25])([CH3:24])[CH3:22]

Participants

Reactant 2

HCID 62493Pivaloyl chloride

HCID 68870563HCID 68870563, compound

Product 1

HCID 57884003HCID 57884003, compound

Procedure

The title compound was prepared according to the procedure described in Step C of Example 17 from 1-({[2-amino-4-(isopropylsulfonyl)phenyl]amino}methyl)cyclopentanol (Step B) and pivaloyl chloride.

Sources & evidence

ORD record: ord-57dcd0a3e9b34827bb8b2f201e76408e
Source dataset: uspto-grants-2009_10
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US07598393B2

Reaction notes

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