HuagongsheHuagongshe Chemistry Print Report · For research reference only
3-Fluorophenylboronic acid → 5-(3-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-2(3H)-one
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 3-Fluorophenylboronic acid | HCID 2733986 | — |
| Reactant | 5-bromo-1H,2H,3H-pyrrolo(2,3-b)pyridin-2-one | HCID 15504062 | — |
| Product | 5-(3-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-2(3H)-one | HCID 46912085 | 32% |
Reaction Steps
The title compound was prepared in 32% yield according to the procedure described in Example 2, starting from 5-bromo-1,3-dihydro-pyrrolo[2,3-b]pyridin-2-one (prepared according to the procedure described in WO2003082868, Page 33) and 3-fluoro-phenyl boronic acid. 1H NMR is the same as the one reported in WO2003082868, page 34.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07608712B2 |
| Source dataset | uspto-grants-2009_10 |
| ORD ID | ord-2a3ffec6f675480492649423f7849e35 |
| Source note | uspto-grants-2009_10 |