3-Pyridinylboronic acid → HCID 23571182, compound
Reaction equation
Br[C:2]1[S:6][C:5]([C:7]2[CH:8]=[CH:9][C:10]3[CH2:17][CH:16]4[C:18]5([CH2:22][N:21]([CH2:23][C:24]([F:27])([F:26])[F:25])[S:20](=[O:29])(=[O:28])[NH:19]5)[CH:13]([CH2:14][CH2:15]4)[CH2:12][C:11]=3[CH:30]=2)=[N:4][CH:3]=1.[N:31]1[CH:36]=[CH:35][CH:34]=[C:33](B(O)O)[CH:32]=1>>[N:31]1[CH:36]=[CH:35][CH:34]=[C:33]([C:2]2[S:6][C:5]([C:7]3[CH:8]=[CH:9][C:10]4[CH2:17][CH:16]5[C:18]6([CH2:22][N:21]([CH2:23][C:24]([F:27])([F:26])[F:25])[S:20](=[O:29])(=[O:28])[NH:19]6)[CH:13]([CH2:14][CH2:15]5)[CH2:12][C:11]=4[CH:30]=3)=[N:4][CH:3]=2)[CH:32]=1Participants
3
Procedure
Prepared using the bromide from Example 36 Step 2 and 3-pyridylboronic acid by the method described for Example 36 Step 3. MS (ES+) 521 ([MH]+).
Workup
- customPrepared
Sources & evidence
- ORD record
- ord-20f221db4d664dc185b90eca955fd6bb
- Source dataset
- uspto-grants-2006_05
- Patent number
- US07041689B2
Reaction notes
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