Pteridine, 4-(methylthio)- → HCID 10271002, compound

HRID 1827194Notes

Reaction equation

HRID 1827194 reaction equation
[CH2:1]([O:8][C:9]([N:11]1[CH2:16][CH2:15][CH:14]([CH2:17][NH2:18])[CH2:13][CH2:12]1)=[O:10])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1.CS[C:21]1[C:30]2[C:25](=[N:26][CH:27]=[CH:28][N:29]=2)[N:24]=[CH:23][N:22]=1>>[CH2:1]([O:8][C:9]([N:11]1[CH2:16][CH2:15][CH:14]([CH2:17][NH:18][C:21]2[C:30]3[C:25](=[N:26][CH:27]=[CH:28][N:29]=3)[N:24]=[CH:23][N:22]=2)[CH2:13][CH2:12]1)=[O:10])[C:2]1[CH:7]=[CH:6][CH:5]=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 249622Pteridine, 4-(methylthio)-2×HCID 219554994-Aminomethyl-1-N-Cbz-piperidine

Product 1

HCID 10271002HCID 10271002, compound

Procedure

EXAMPLE 86 was prepared from 4-aminomethyl-piperidine-1-carboxylic acid benzyl ester and 4-methylthio-pteridine (4-methylthio-pteridine was prepared according to A. A. Brown, D. J. Brown,h. C. S. Wood, J. Chem. Soc., 1954, 3832–3839): MS (m+1)=379.

Workup

  1. customwas prepared

Sources & evidence

ORD record
ord-9f37f55dedb54af89ad03618140fbdef
Source dataset
uspto-grants-2006_05
Patent number
US07053089B2

Reaction notes

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