Benzo(d)thiazol-2-amine → HCID 22063782, compound

HRID 1828455Notes

Reaction equation

HRID 1828455 reaction equation
[C:1]([C:5]1[N:6]=[C:7]([NH:10][C:11]([C:13]2[CH:28]=[CH:27][N:16]3[C:17](=[O:26])[C:18]([C:21]4[N:22]=[N:23][NH:24][N:25]=4)=[CH:19][N:20]=[C:15]3[CH:14]=2)=[O:12])[S:8][CH:9]=1)(C)(C)[CH3:2].CO[C:31]1C=CC(CN2N=NC(C3C(=O)N4C=CC(C(O)=O)=CC4=NC=3)=N2)=C[CH:32]=1.NC1SC2C=CC=CC=2N=1>>[S:8]1[C:9]2[CH:31]=[CH:32][CH:2]=[CH:1][C:5]=2[N:6]=[C:7]1[NH:10][C:11]([C:13]1[CH:28]=[CH:27][N:16]2[C:17](=[O:26])[C:18]([C:21]3[N:25]=[N:24][NH:23][N:22]=3)=[CH:19][N:20]=[C:15]2[CH:14]=1)=[O:12]

Participants

4

Reactant 3

HCID 8706Benzo(d)thiazol-2-amineHCID 22063508HCID 22063508, compoundHCID 22063552HCID 22063552, compound

Product 1

HCID 22063782HCID 22063782, compound

Procedure

Reactions were performed in the same manner as in Example 10, (F) by using 3-[2-(4-methoxybenzyl)-2H-1,2,3,4-tetrazol-5-yl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-8-carboxylic acid (60 mg, 0.16 mmol) and 2-aminobenzothiazole (30 mg, 0.17 mmol) to obtain 2 mg (3% for the two steps) of an orange compound.

Workup

  1. customto obtain 2 mg (3% for the two steps) of an orange compound

Sources & evidence

ORD record
ord-b62b8882289c4031a65c91db0c8bd9e9
Source dataset
uspto-grants-2006_06
Patent number
US07056917B2

Reaction notes

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