HCID 12226750, compound → HCID 12226751, compound

HRID 1833555Notes

Reaction equation

HRID 1833555 reaction equation
CN1CC[N:5]([C:8](=[O:25])[CH2:9][C:10]2([CH3:24])[C:15]3=[C:16]([CH3:23])[C:17]4[CH:18]=[CH:19][CH:20]=[CH:21][C:22]=4[N:14]3[CH2:13][CH2:12][O:11]2)[CH2:4][CH2:3]1.CNC(=O)CC1(C)C2=C(C)C3C=CC=CC=3N2CCO1>>[CH3:24][C:10]1([CH2:9][C:8]([NH:5][CH2:4][CH3:3])=[O:25])[C:15]2=[C:16]([CH3:23])[C:17]3[CH:18]=[CH:19][CH:20]=[CH:21][C:22]=3[N:14]2[CH2:13][CH2:12][O:11]1

Participants

3

Reactant 2

HCID 12226750HCID 12226750, compoundHCID 12226762HCID 12226762, compound

Product 1

HCID 12226751HCID 12226751, compound

Procedure

By following the procedure of Example 284 but using as starting material an equivalent amount of one of the amide compounds of formula V, described in Examples 108 to 283 instead of N,1,10-trimethyl-3,4-dihydro-1H-1,4-oxazino[4,3-a]indole-1-acetamide, then the corresponding compounds of formula I are obtained. Examples of such compounds of formula I are listed as products in Tables VII and VIII together with the appropriate starting material. In each case the starting material is noted by the example in which it is prepared.

Workup

  1. customthe corresponding compounds of formula I are obtained
  2. customis prepared

Sources & evidence

ORD record
ord-243e7466a41441ad9a3e7a97d55dfadf
Source dataset
uspto-grants-1978_01
Patent number
US04066763

Reaction notes

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