Back
HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 18434Generated: October 25, 2026

3-(N,N-Dimethylsulphonamido)benzeneboronic acid → 3-(2-{[dihydroxy(1-methylethyl)-lambda4-sulfanyl]amino}-2,3-dihydro-1H-inden-5-yl)-N,N-dimethylbenzenesulfonamide

https://huagongshe.com/reaction/18434

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-(N,N-Dimethylsulphonamido)benzeneboronic acidHCID 44119634—
ReactantN-(5-iodo-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamideHCID 46899809—
Product3-(2-{[dihydroxy(1-methylethyl)-lambda4-sulfanyl]amino}-2,3-dihydro-1H-inden-5-yl)-N,N-dimethylbenzenesulfonamideHCID 68447569—

Reaction Steps

The title compound was prepared from N-(5-iodo-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide and {3-[(dimethylamino)sulfonyl]phenyl}boronic acid (WO2003004472) in a similar manner to Example 1.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07741351B2
Source datasetuspto-grants-2010_06
ORD IDord-42b9c346e4594c3b87f17142402350a2
Source noteuspto-grants-2010_06