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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 18435Generated: October 25, 2026

3-(Aminosulphonyl)benzeneboronic acid → 3-(2-{[dihydroxy(1-methylethyl)-lambda4-sulfanyl]amino}-2,3-dihydro-1H-inden-5-yl)benzenesulfonamide

https://huagongshe.com/reaction/18435

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-(Aminosulphonyl)benzeneboronic acidHCID 44119323—
ReactantN-(5-iodo-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamideHCID 46899809—
Product3-(2-{[dihydroxy(1-methylethyl)-lambda4-sulfanyl]amino}-2,3-dihydro-1H-inden-5-yl)benzenesulfonamideHCID 68446923—

Reaction Steps

The title compound was prepared from N-(5-iodo-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide and [3-(aminosulfonyl)phenyl]boronic acid (WO2003004472) in a similar manner to Example 1.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07741351B2
Source datasetuspto-grants-2010_06
ORD IDord-92d8d03154da4df1bf9554108293e953
Source noteuspto-grants-2010_06