Participants
| Role | Name | HCID | Charge |
|---|
| Reactant | Oxalyl chloride | HCID 65578 | — |
| Reactant | 5-Ethyl-1,3,4-oxadiazol-2-amine | HCID 343487 | — |
| Reactant | Potassium bisulfate | HCID 516920 | — |
| Reactant | HCID 86200989 | HCID 86200989 | — |
| Catalyst | 4-(Dimethylamino)pyridine | HCID 14284 | — |
| Solvent | Water | HCID 962 | — |
| Solvent | Pyridine | HCID 1049 | — |
| Solvent | Dimethylformamide | HCID 6228 | — |
| Product | HCID 89545072 | HCID 89545072 | — |
Reaction Steps
400 mg (1.61 mmol) of 2,4-dichloro-3-[(methoxyimino)methyl]benzoic acid and 228 mg (2.0 mmol) of 5-ethyl-1,3,4-oxadiazole-2-amine were dissolved in 3 ml of pyridine, and 10 mg of 4-dimethylaminopyridine and a drop of DMF were added. At room temperature (RT), 255.83 mg (2.016 mmol) of oxalyl chloride were then added dropwise, and the mixture was stirred at 70° C. for 4 h. 0.5 ml of water was then added to the reaction, which had once more been cooled, and the mixture was stirred for about 30 min, acidified with a saturated KHSO4 solution and extracted three times with in each case 100 ml of ethyl acetate. The combined organic phases were washed once with 20 ml of a saturated NaHCO3 solution, dried over MgSO4, filtered off and concentrated. The residue was purified chromatographically by preparative HPLC. Yield: 99.3 mg (18%) as colorless crystals.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
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| Patent number | US08957096B2 |
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| Source dataset | uspto-grants-2015_02 |
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| ORD ID | ord-112c55b5d7c74960a1e0cd20742b360c |
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| Source note | uspto-grants-2015_02 |
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