4-Aminobenzylamine → HCID 86674541, compound
Reaction equation
[NH2:1][C:2]1[CH:9]=[CH:8][C:5]([CH2:6][NH2:7])=[CH:4][CH:3]=1.C([O:14][C:15]([C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][C:18]=1[C:23]1[CH:28]=[CH:27][C:26]([CH2:29][N:30]2[C:38]3[C:33](=[CH:34][C:35]([C:39](O)=[O:40])=[CH:36][CH:37]=3)[C:32]([CH3:42])=[C:31]2[CH3:43])=[CH:25][CH:24]=1)=[O:16])(C)(C)C>>[NH2:1][C:2]1[CH:9]=[CH:8][C:5]([CH2:6][NH:7][C:39]([C:35]2[CH:34]=[C:33]3[C:38](=[CH:37][CH:36]=2)[N:30]([CH2:29][C:26]2[CH:25]=[CH:24][C:23]([C:18]4[C:17]([C:15]([OH:16])=[O:14])=[CH:22][CH:21]=[CH:20][CH:19]=4)=[CH:28][CH:27]=2)[C:31]([CH3:43])=[C:32]3[CH3:42])=[O:40])=[CH:4][CH:3]=1Participants
3
Procedure
The title compound was prepared following the same general protocol as described in Steps 8-9, Example 1, using 4-aminobenzylamine and 1-((2′-(tert-butoxycarbonyl)biphenyl-4-yl)methyl)-2,3-dimethyl-1H-indole-5-carboxylic acid.
Sources & evidence
- ORD record
- ord-af92047279a04be885719bc7138e1ff0
- Source dataset
- uspto-grants-2015_02
- Patent number
- US08957093B2
Reaction notes
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