9-bromo-8-methoxy-6-methylthieno[2,3-c]quinolin-4(5H)-one → HCID 86689455, compound

Participants

Reaction Steps

Following General Procedure B, 9-bromo-8-methoxy-6-methylthieno[2,3-c]quinolin-4(5H)-one) (900 mg, 2.9 mmol) was reacted with (R)-tert-butyl 2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)butylcarbamate (900 mg, 2.7 mmol) to afford the desired product (190 mg, 15%) as a yellow solid: ESI MS m % z 493 [C28H32N2O4S+H]+.

Provenance & Evidence