N-Ethylaniline → ethyl 3-(4-benzyloxyphenyl)-2-(phenyl-N-ethylamino)propionate

Participants

Reaction Steps

In a similar manner to that described in Reference example 55(a), a reaction was carried out using ethyl 3-(4-benzyloxyphenyl)-2-methanesulfonyloxypropionate (4.50 g) and N-ethylaniline (5.6 ml) and the reaction mixture was treated to afford a mixture of the desired compound and N-ethylaniline (6.30 g) as a syrup.

Provenance & Evidence