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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1867813Generated: October 30, 2026

(6-Methoxypyridin-3-yl)boronic acid → [4-(6-Methoxy-pyridin-3-yl)-phenyl]-(2-(S)-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-methanone

https://huagongshe.com/reaction/1867813

Reaction equation

Participants

RoleNameHCIDCharge
Reactant(6-Methoxypyridin-3-yl)boronic acidHCID 2734368—
ReactantPyrrolidine, 1-(4-bromobenzoyl)-2-(1-pyrrolidinylmethyl)-, (2S)-HCID 11965129—
Product[4-(6-Methoxy-pyridin-3-yl)-phenyl]-(2-(S)-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-methanoneHCID 57980121—

Reaction Steps

The title compound is prepared in a manner substantially analogous to Procedure SS starting from 2-Methoxy-5-pyridine boronic acid and (4-bromo-phenyl)-(2-(S)-pyrrolidin-1-ylmethyl-pyrrolidin-1-yl)-methanone. MS (ES+) 366.4

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07632857B2
Source datasetuspto-grants-2009_12
ORD IDord-8b3618a9e9da44df8fa771b5635be191
Source noteuspto-grants-2009_12