3-Amino-3-methylbutanamide → 4-[(4-{3-[2-Carbamoyl-1,1-di(methyl)ethylamino]propoxy}-2-methylphenyl)methyl]-3-(beta-D-galactopyranosyloxy)-5-isopropyl-1H-pyrazole

Participants

Reaction Steps

The title compound was prepared in a similar manner to that described in Example 72 using 3-(2,3,4,6-tetra-O-acetyl-β-D-galactopyranosyloxy)-4-{[4-(3-hydroxypropoxy)-2-methylphenyl]methyl}-5-isopropyl-1H-pyrazole and 3-amino-3-methylbutyramide instead of 3-(2,3,4,6-tetra-O-acetyl-β-D-glucopyranosyloxy)-4-{[4-(3-hydroxypropoxy)phenyl]-methyl}-5-isopropyl-1H-pyrazole and 2-[2-amino-2-(methyl)-propionylamino]ethanol, respectively.

Provenance & Evidence