反应详情

The title compound was prepared from 1-acetyl-5-bromo-6-[(1-methyl-1,2,5,6-tetrahydropyridine-4-yl)methoxy]indoline (D65) using a similar procedure to Description 8b in WO96/19477, but with toluene at 80° C. in place of refluxing benzene. The product was obtained from the acid/base purification as a beige solid (94%).

1. customat 80° C.