1-[4-(Bromomethyl)phenyl]-1H-pyrrole → HCID 24956848, compound

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The title compound was prepared from 4-methyl-2-(2H-pyrazol-3-yl)-thiazole-5-carboxylic acid (pyridin-3-ylmethyl)-amide and 1-(4-bromomethyl-phenyl)-1H-pyrrole as described in Example 49 and isolated as a white solid (0.08 g, 52% yield). 1H NMR (400 MHz, CDCl3) δ 8.60 (s, 1H), 8.54-8.57 (m, 1H), 7.71 (d, J=8.1 Hz, 1H), 7.26-7.43 (m, 6H), 7.07 (d, J=8 Hz, 2H), 6.86 (s, 1H), 6.35 (d, J=4 Hz, 2H), 6.18-6.25 (m, 1H), 5.36 (s, 2H), J=8 Hz, 2H), 2.75 (s, 3H); MS (M+H)+=455.2; Rt=1.38 min; HRMS (M+H)+=455.17.

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