1-(Bromomethyl)-4-(trifluoromethoxy)benzene → HCID 24951858, compound

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The title compound was prepared from 4-methyl-2-(2H-pyrazol-3-yl)-thiazole-5-carboxylic acid (pyridin-3-ylmethyl)-amide and bromomethyl-4-trifluoromethoxy-benzene as described in Example 49 and isolated as a yellow solid (0.078 g, 52% yield) 1H NMR (400 MHz, CDCl3) δ 8.61 (s, 1H), 8.56 (d, J=4 Hz, 1H), 7.71 (d, J=8 Hz, 1H), 7.41 (d, J=2 Hz, 1H), 7.26-7:31 (m, 3H), 7.17-7.23 (m, 2H), 6.86 (d, J=2 Hz, 1H), 6.10-6.16 (m, 1H), 5.35 (s, 2H), 4.63 (d, J=8 Hz, 2H), 2.75 (s, 3H); MS (M+H)+=474.1; Rt=1.38 min; HRMS (M+H)+=474.12.

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