3,5-Dimethylphenylboronic acid → HCID 178425110, compound

HRID 1890297Notes

Reaction equation

HRID 1890297 reaction equation
C([O:8][C:9]1[N:14]=[C:13]2[NH:15][CH:16]=[N:17][C:12]2=[CH:11][CH:10]=1)C1C=CC=CC=1.[CH3:18][C:19]1[CH:20]=[C:21](B(O)O)[CH:22]=[C:23]([CH3:25])[CH:24]=1>>[CH3:18][C:19]1[CH:20]=[C:21]([N:15]2[C:13]3=[N:14][C:9]([OH:8])=[CH:10][CH:11]=[C:12]3[N:17]=[CH:16]2)[CH:22]=[C:23]([CH3:25])[CH:24]=1

Participants

3

Reactant 2

HCID 27343493,5-Dimethylphenylboronic acidHCID 178420377HCID 178420377, compound

Product 1

HCID 178425110HCID 178425110, compound

Procedure

From 5-(benzyloxy)-3H-imidazo[4,5-b]pyridine and 3,5-dimethylphenylboronic acid, prepared in a similar manner as the one described in Example 1.26, the title compound was obtained. LCMS m/z=239.9 [M+H]+.

Sources & evidence

ORD record
ord-4c97bdeca9614d5381bf307f0dff0904
Source dataset
uspto-grants-2013_08
Patent number
US08507473B2

Reaction notes

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