Thiophene-3-boronic acid → HCID 178515774, compound

HRID 1890299Notes

Reaction equation

HRID 1890299 reaction equation
C([O:8][C:9]1[N:14]=[C:13]2[NH:15][CH:16]=[N:17][C:12]2=[CH:11][CH:10]=1)C1C=CC=CC=1.[S:18]1[CH:22]=[CH:21][C:20](B(O)O)=[CH:19]1>>[S:18]1[CH:22]=[CH:21][C:20]([N:15]2[C:13]3=[N:14][C:9]([OH:8])=[CH:10][CH:11]=[C:12]3[N:17]=[CH:16]2)=[CH:19]1

Participants

3

Reactant 2

HCID 581760Thiophene-3-boronic acidHCID 178420377HCID 178420377, compound

Product 1

HCID 178515774HCID 178515774, compound

Procedure

From 5-(benzyloxy)-3H-imidazo[4,5-b]pyridine and thiophen-3-ylboronic acid, prepared in a similar manner as the one described in Example 1.26, the title compound was obtained. LCMS m/z=218.1 [M+H]+.

Sources & evidence

ORD record
ord-de15e38508e3426a8f246ee8b95669e5
Source dataset
uspto-grants-2013_08
Patent number
US08507473B2

Reaction notes

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