2-Ethylphenylboronic Acid (contains varying amounts of Anhydride) → HCID 178436073, compound

HRID 1890307Notes

Reaction equation

HRID 1890307 reaction equation
C([O:8][C:9]1[N:14]=[C:13]2[NH:15][CH:16]=[N:17][C:12]2=[CH:11][CH:10]=1)C1C=CC=CC=1.[CH2:18]([C:20]1[CH:25]=[CH:24][CH:23]=[CH:22][C:21]=1B(O)O)[CH3:19]>>[CH2:18]([C:20]1[CH:25]=[CH:24][CH:23]=[CH:22][C:21]=1[N:15]1[C:13]2=[N:14][C:9]([OH:8])=[CH:10][CH:11]=[C:12]2[N:17]=[CH:16]1)[CH3:19]

Participants

3

Reactant 2

HCID 41008622-Ethylphenylboronic Acid (contains varying amounts of Anhydride)HCID 178420377HCID 178420377, compound

Product 1

HCID 178436073HCID 178436073, compound

Procedure

From 5-(benzyloxy)-3H-imidazo[4,5-b]pyridine and 2-ethylphenylboronic acid, prepared in a similar manner as the one described in Example 1.26, the title compound was obtained. LCMS m/z=239.9 [M+H]+.

Sources & evidence

ORD record
ord-8f28d8f0e81e42559c3ac6a89d485d43
Source dataset
uspto-grants-2013_08
Patent number
US08507473B2

Reaction notes

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