HCID 68597910, compound → HCID 68597678, compound

HRID 1890379Notes

Reaction equation

HRID 1890379 reaction equation
[NH:1]1[C:9]2[C:4](=[CH:5][C:6]([CH:10]3[CH2:13][N:12]([C:14]([O:16][C:17]([CH3:20])([CH3:19])[CH3:18])=[O:15])[CH2:11]3)=[CH:7][CH:8]=2)[CH:3]=[N:2]1.[F:21][C:22]1[CH:27]=[CH:26][C:25]([S:28](Cl)(=[O:30])=[O:29])=[CH:24][C:23]=1[C:32]1[N:33]=[CH:34][O:35][CH:36]=1>>[F:21][C:22]1[CH:27]=[CH:26][C:25]([S:28]([N:1]2[C:9]3[C:4](=[CH:5][C:6]([CH:10]4[CH2:13][N:12]([C:14]([O:16][C:17]([CH3:20])([CH3:19])[CH3:18])=[O:15])[CH2:11]4)=[CH:7][CH:8]=3)[CH:3]=[N:2]2)(=[O:30])=[O:29])=[CH:24][C:23]=1[C:32]1[N:33]=[CH:34][O:35][CH:36]=1

Participants

3

Reactant 2

HCID 68597910HCID 68597910, compoundHCID 86642048HCID 86642048, compound

Product 1

HCID 68597678HCID 68597678, compound

Procedure

This compound was prepared from tert-butyl 3-(1H-indazol-5-yl)azetidine-1-carboxylate and 4-fluoro-3-(oxazol-4-yl)benzene-1-sulfonyl chloride by analogy to the method outlined in example 44.c, below).

Sources & evidence

ORD record
ord-6a0b60b5b74547adbc6848ad2bd20a33
Source dataset
uspto-grants-2013_08
Patent number
US08507469B2

Reaction notes

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