Tert-butyl 3-oxopiperidine-1-carboxylate → HCID 59799765, compound

HRID 1911908Notes

Reaction equation

HRID 1911908 reaction equation
O=[C:2]1[CH2:7][CH2:6][CH2:5][N:4]([C:8]([O:10][C:11]([CH3:14])([CH3:13])[CH3:12])=[O:9])[CH2:3]1.[NH2:15][C:16]1[CH:21]=[CH:20][C:19]([C:22]2[C:23]([NH2:27])=[N:24][O:25][N:26]=2)=[CH:18][CH:17]=1>>[NH2:27][C:23]1[C:22]([C:19]2[CH:20]=[CH:21][C:16]([NH:15][CH:2]3[CH2:7][CH2:6][CH2:5][N:4]([C:8]([O:10][C:11]([CH3:14])([CH3:13])[CH3:12])=[O:9])[CH2:3]3)=[CH:17][CH:18]=2)=[N:26][O:25][N:24]=1

Participants

3

Reactant 2

HCID 2756825Tert-butyl 3-oxopiperidine-1-carboxylateHCID 59799786HCID 59799786, compound

Product 1

HCID 59799765HCID 59799765, compound

Procedure

Reaction of tert-butyl 3-oxopiperidine-1-carboxylate and 4-(4-aminophenyl)-1,2,5-oxadiazol-3-amine using the method of Example 3 afforded the title compound.

Sources & evidence

ORD record
ord-e52f5a1aabdf4cbab03b63cebeb191e0
Source dataset
uspto-grants-2013_12
Patent number
US08604205B2

Reaction notes

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