2-Methoxypyrimidine-5-boronic acid → 2-(4-fluorophenyl)-N-[3-(2-methoxypyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-2-yl]acetamide

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Reaction Steps

The product from Example 140A and 2-methoxypyrimidine-5-boronic acid were processed using the method analogous to that described in Example 110C to provide the title compound. 1H NMR (400 MHz, DMSO-d6) δ ppm 10.69-10.71 (m, 1H), 9.12 (dd, J=6.9, 1.7 Hz, 1H), 8.74 (s, 2H), 8.62 (dd, J=4.1, 1.7 Hz, 1H), 7.30-7.35 (m, 2H), 7.12-7.17 (m, 3H), 3.94 (s, 3H), 3.69 (s, 2H); MS (ESI) m/z 379 (M+H)+.

Provenance & Evidence