2-Methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenylamine → HCID 59401757, compound

HRID 1916937Notes

Reaction equation

HRID 1916937 reaction equation
[CH3:1][C:2]1[CH:7]=[C:6]([N:8]2[CH2:12][CH2:11][CH:10]([N:13]3[CH2:17][CH2:16][CH2:15][CH:14]3[CH3:18])[CH2:9]2)[CH:5]=[CH:4][C:3]=1[NH2:19].[C:20]([N:23]1[CH2:28][CH2:27][CH2:26][CH:25]([C:29]2[CH:37]=[CH:36][C:32]([C:33](O)=[O:34])=[CH:31][CH:30]=2)[CH2:24]1)(=[O:22])[CH3:21]>>[C:20]([N:23]1[CH2:28][CH2:27][CH2:26][CH:25]([C:29]2[CH:30]=[CH:31][C:32]([C:33]([NH:19][C:3]3[CH:4]=[CH:5][C:6]([N:8]4[CH2:12][CH2:11][CH:10]([N:13]5[CH2:17][CH2:16][CH2:15][CH:14]5[CH3:18])[CH2:9]4)=[CH:7][C:2]=3[CH3:1])=[O:34])=[CH:36][CH:37]=2)[CH2:24]1)(=[O:22])[CH3:21]

Participants

3

Reactant 2

HCID 594018302-Methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenylamineHCID 67401293HCID 67401293, compound

Product 1

HCID 59401757HCID 59401757, compound

Procedure

The title compound was prepared in a manner substantially the same as example 1 by coupling 2-methyl-4-(2-methyl-[1,3′]bipyrrolidinyl-1′-yl)-phenylamine with 4-(1-acetyl-piperidin-3-yl)-benzoic acid. MS: 489.3 (M+H).

Sources & evidence

ORD record
ord-977a7cb507c84745905fa5f0aa0597db
Source dataset
uspto-grants-2013_12
Patent number
US08618159B2

Reaction notes

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