1-(Propan-2-yl)-1H-benzotriazole-5-carboxylic acid → HCID 59401829, compound

HRID 1916955Notes

Reaction equation

HRID 1916955 reaction equation
[CH3:1][C:2]1[CH:7]=[C:6]([N:8]2[CH2:12][CH2:11][CH:10]([N:13]3[CH2:17][CH2:16][CH2:15][CH:14]3[CH3:18])[CH2:9]2)[CH:5]=[CH:4][C:3]=1[NH2:19].[CH:20]([N:23]1[C:27]2[CH:28]=[CH:29][C:30]([C:32](O)=[O:33])=[CH:31][C:26]=2[N:25]=[N:24]1)([CH3:22])[CH3:21]>>[CH3:1][C:2]1[CH:7]=[C:6]([N:8]2[CH2:12][CH2:11][CH:10]([N:13]3[CH2:17][CH2:16][CH2:15][CH:14]3[CH3:18])[CH2:9]2)[CH:5]=[CH:4][C:3]=1[NH:19][C:32]([C:30]1[CH:29]=[CH:28][C:27]2[N:23]([CH:20]([CH3:21])[CH3:22])[N:24]=[N:25][C:26]=2[CH:31]=1)=[O:33]

Participants

3

Reactant 2

HCID 27366901-(Propan-2-yl)-1H-benzotriazole-5-carboxylic acidHCID 594018302-Methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenylamine

Product 1

HCID 59401829HCID 59401829, compound

Procedure

The title compound was prepared in a manner substantially the same as example 1 by coupling 2-methyl-4-(2-methyl-[1,3′]bipyrrolidinyl-1′-yl)-phenylamine with 1-isopropyl-1H-benzotriazole-5-carboxylic acid. MS: 447.3 (M+H).

Sources & evidence

ORD record
ord-f1d23bd12880423a9d1888e3f233614c
Source dataset
uspto-grants-2013_12
Patent number
US08618159B2

Reaction notes

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