1H-indole-6-carboxylic acid → HCID 59401827, compound

HRID 1916958Notes

Reaction equation

HRID 1916958 reaction equation
[CH3:1][C:2]1[CH:7]=[C:6]([N:8]2[CH2:12][CH2:11][CH:10]([N:13]3[CH2:17][CH2:16][CH2:15][CH:14]3[CH3:18])[CH2:9]2)[CH:5]=[CH:4][C:3]=1[NH2:19].[NH:20]1[C:28]2[C:23](=[CH:24][CH:25]=[C:26]([C:29](O)=[O:30])[CH:27]=2)[CH:22]=[CH:21]1>>[CH3:1][C:2]1[CH:7]=[C:6]([N:8]2[CH2:12][CH2:11][CH:10]([N:13]3[CH2:17][CH2:16][CH2:15][CH:14]3[CH3:18])[CH2:9]2)[CH:5]=[CH:4][C:3]=1[NH:19][C:29]([C:26]1[CH:27]=[C:28]2[C:23]([CH:22]=[CH:21][NH:20]2)=[CH:24][CH:25]=1)=[O:30]

Participants

3

Reactant 2

HCID 5952301H-indole-6-carboxylic acidHCID 594018302-Methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenylamine

Product 1

HCID 59401827HCID 59401827, compound

Procedure

The title compound was prepared in a manner substantially the same as example 1 by coupling 2-methyl-4-(2-methyl-[1,3′]bipyrrolidinyl-1′-yl)-phenylamine with 1H-indole-6-carboxylic acid. MS: 403.3 (M+H).

Sources & evidence

ORD record
ord-ea7fc736463d4cb391df443596d84160
Source dataset
uspto-grants-2013_12
Patent number
US08618159B2

Reaction notes

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