4-(1-Pyrrolidinyl)piperidine → HCID 58808605, compound

HRID 1921472Notes

Reaction equation

HRID 1921472 reaction equation
[CH2:1]([C:3]1[C:8](=[O:9])[NH:7][C:6]([CH3:10])=[C:5]([C:11]2[CH:16]=[CH:15][CH:14]=[C:13]([CH:17]=O)[N:12]=2)[CH:4]=1)[CH3:2].[N:19]1([CH:24]2[CH2:29][CH2:28][NH:27][CH2:26][CH2:25]2)[CH2:23][CH2:22][CH2:21][CH2:20]1>>[CH2:1]([C:3]1[C:8](=[O:9])[NH:7][C:6]([CH3:10])=[C:5]([C:11]2[CH:16]=[CH:15][CH:14]=[C:13]([CH2:17][N:27]3[CH2:28][CH2:29][CH:24]([N:19]4[CH2:23][CH2:22][CH2:21][CH2:20]4)[CH2:25][CH2:26]3)[N:12]=2)[CH:4]=1)[CH3:2]

Participants

3

Reactant 2

HCID 787034-(1-Pyrrolidinyl)piperidineHCID 58808670HCID 58808670, compound

Product 1

HCID 58808605HCID 58808605, compound

Procedure

5′-Ethyl-2′-methyl-6′-oxo-1′,6′-dihydro-[2,3′]bipyridinyl-6-carbaldehyde prepared in accordance with PREPARATION 11 is reacted with 4-pyrrolidinyl-piperidine as described in Method A, Example 123 to give the title compound. MS: m/e=381 (M+H).

Sources & evidence

ORD record
ord-f521a76438054ec8bcb8d9edead3c445
Source dataset
uspto-grants-2012_05
Patent number
US08173682B2

Reaction notes

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