Benzoic acid, 4-(phenylsulfonyl)- → HCID 11842650, compound

HRID 1923476Notes

Reaction equation

HRID 1923476 reaction equation
[C:1]1([S:7]([C:10]2[CH:18]=[CH:17][C:13]([C:14]([OH:16])=O)=[CH:12][CH:11]=2)(=[O:9])=[O:8])[CH:6]=[CH:5][CH:4]=[CH:3][CH:2]=1.[NH:19]1[CH2:23][CH2:22][CH2:21][C@H:20]1[CH2:24][N:25]1[CH2:29][CH2:28][CH2:27][CH2:26]1>>[C:1]1([S:7]([C:10]2[CH:11]=[CH:12][C:13]([C:14]([N:19]3[CH2:23][CH2:22][CH2:21][C@H:20]3[CH2:24][N:25]3[CH2:29][CH2:28][CH2:27][CH2:26]3)=[O:16])=[CH:17][CH:18]=2)(=[O:8])=[O:9])[CH:2]=[CH:3][CH:4]=[CH:5][CH:6]=1

Participants

3

Reactant 2

HCID 79322Benzoic acid, 4-(phenylsulfonyl)-HCID 853152(S)-(+)-1-(2-Pyrrolidinylmethyl)pyrrolidine

Product 1

HCID 11842650HCID 11842650, compound

Procedure

The title compound is prepared in a manner substantially analogous to the procedures found in Intermediate 6 and Example 17 using 4-(phenylsulfonyl)-benzoic acid [CAS# 5361-54-6] and (S)-(+)-1-(2-pyrrolidinylmethyl)pyrrolidine.

Sources & evidence

ORD record
ord-0492c9fabecf4f73899d881d3905ee57
Source dataset
uspto-grants-2012_05
Patent number
US08178528B2

Reaction notes

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